Ident. | Authors (with country if any) | Title |
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000A38 |
Emilia Bankowska [Pologne] ; Jan Balzarini [Belgique] ; Iwona E. Głowacka [Pologne] ; Andrzej E. Wr Blewski [Pologne] | Design, synthesis, antiviral and cytotoxic evaluation of novel acyclic phosphonate nucleotide analogues with a 5,6-dihydro-1H-[1,2,3]triazolo[4,5-d]pyridazine-4,7-dione system |
000A56 |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Novel Acyclic Phosphonylated 1,2,3‐Triazolonucleosides with an Acetamidomethyl Linker: Synthesis and Biological Activity |
000A62 |
Magdalena Łysakowska [Pologne] ; Jan Balzarini [Belgique] ; Dorota G. Piotrowska [Pologne] | Design, Synthesis, Antiviral, and Cytostatic Evaluation of Novel Isoxazolidine Analogs of Homonucleotides |
000A68 |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Dorota G. Piotrowska [Pologne] | 1‐Amino‐3‐(1H‐1,2,3‐triazol‐1‐yl)propylphosphonates as Acyclic Analogs of Nucleotides |
000B09 |
Christopher Mcguigan [Royaume-Uni] ; Claire Bourdin [Royaume-Uni] ; Marco Derudas [Royaume-Uni] ; Nadège Hamon [Royaume-Uni] ; Karen Hinsinger [Royaume-Uni] ; Sahar Kandil [Royaume-Uni] ; Karolina Madela [Royaume-Uni] ; Silvia Meneghesso [Royaume-Uni] ; Fabrizio Pertusati [Royaume-Uni] ; Michaela Serpi [Royaume-Uni] ; Magdalena Slusarczyk [Royaume-Uni] ; Stanley Chamberlain [États-Unis] ; Alexander Kolykhalov [États-Unis] ; John Vernachio [États-Unis] ; Christophe Vanpouille [États-Unis] ; Andrea Introini [États-Unis] ; Leonid Margolis [États-Unis] ; Jan Balzarini [Belgique] | Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides |
000B26 |
Rosa Miralles-Llumà [Espagne] ; Antoni Figueras [Espagne] ; Félix Busqué [Espagne] ; Angel Alvarez-Larena [Espagne] ; Jan Balzarini [Belgique] ; Marta Figueredo [Espagne] ; Josep Font [Espagne] ; Ramon Alibés [Espagne, Canada] ; Jean-Didier Maréchal [Espagne, Canada] | Synthesis, Antiviral Evaluation, and Computational Studies of Cyclobutane and Cyclobutene L‐Nucleoside Analogues |
000B27 |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Synthesis of a New Series of Phosphonylated 1,2,3‐Triazoles as Acyclic Analogs of Ribavirin |
000B28 |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Synthesis and Biological Evaluation of Novel 1,2,3‐Triazolonucleotides |
000B54 |
Mahesh K. Lakshman [États-Unis] ; Amit Kumar [États-Unis] ; Raghavan Balachandran [États-Unis] ; Billy W. Day [États-Unis] ; Graciela Andrei [Belgique] ; Robert Snoeck [Belgique] ; Jan Balzarini [Belgique] | Synthesis and Biological Properties of C-2 Triazolylinosine Derivatives |
000B99 |
Subhas S. Karki [Inde] ; Amol A. Kulkarni [Inde] ; Sujeet Kumar [Inde] ; Suresh Kumar Veliyath [Inde] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] | Synthesis and biological evaluation of 2-(5-substituted-1-((diethylamino)methyl)-2-oxoindolin-3-ylidene)- N -substituted-hydrazinecarbothioamides |
000C25 |
Kazuhiro Haraguchi [Japon] ; Hisashi Shimada [Japon] ; Keigo Kimura [Japon] ; Genta Akutsu [Japon] ; Hiromichi Tanaka [Japon] ; Hiroshi Abe [Japon] ; Takayuki Hamasaki [Japon] ; Masanori Baba [Japon] ; Elizabeth A. Gullen [États-Unis] ; Ginger E. Dutschman [États-Unis] ; Yung-Chi Cheng [États-Unis] ; Jan Balzarini [Belgique] | Synthesis of 4′-Ethynyl-2′-deoxy-4′-thioribonucleosides and Discovery of a Highly Potent and Less Toxic NRTI |
000C56 |
Lawrence P. Tardibono [États-Unis] ; Marvin J. Miller [États-Unis] ; Jan Balzarini [Belgique] | Enantioselective syntheses of carbocyclic nuleosides 5′-homocarbovir, epi-4′-homocarbovir and their cyclopropylamine analogs using facially selective Pd-mediated allylations |
000C64 |
Davorka Završnik ; Samija Muratovi ; Damjan Makuc [Slovénie] ; Janez Plavec [Slovénie] ; Mario Cetina [Croatie] ; Ante Nagl [Croatie] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] ; Mladen Mintas [Croatie] | Benzylidene-bis-(4-Hydroxycoumarin) and Benzopyrano-Coumarin Derivatives: Synthesis, 1H/13C-NMR Conformational and X-ray Crystal Structure Studies and In Vitro Antiviral Activity Evaluations |
000C68 |
Alamelu Mahalingam [États-Unis] ; Anthony R. Geonnotti [États-Unis] ; Jan Balzarini [Belgique] ; Patrick F. Kiser [États-Unis] | Activity and Safety of Synthetic Lectins Based on Benzoboroxole-Functionalized Polymers for Inhibition of HIV Entry |
000E60 |
Ivana Perkovi [Croatie] ; Ivan Butula [Croatie] ; Branka Zorc [Croatie] ; Karlo Hock [Croatie] ; Sandra Kraljevi Paveli [Croatie] ; Krešimir Paveli [Croatie] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] ; Mladen Mintas [Croatie] | Novel Lipophilic Hydroxyurea Derivatives: Synthesis, Cytostatic and Antiviral Activity Evaluations |